Solubility: Soluble in DMSO (up to 25 mg/ml) or in Ethanol (up to 25 mg/ml).
Storage: -20°C
Stability: ≥ 2 years.
Applications
GPR55 agonist; endogenous cannabinoid
Functions
Endogenous cannabinoid. Weak ligand for CB1 (Ki=23.8 µM) and CB2 (Ki=13.9 µM) receptor. Selective agonist at GPR55. Inhibits expression of fatty acid amide hydrolase (FAAH). Displays immunosuppressant and anti-inflammatory activity and reduces granuloma-induced hyperalgesia.
Application Procedures
First dissolved in DMSO (up to 25 mg/ml) or in Ethanol (up to 25 mg/ml), then diluted to aqueous buffer. Solutions in water may be stored at -20°C for up to 3 months.
